Impact of Target Warhead and Linkage Vector on Inducing Protein Degradation: Comparison of Bromodomain and Extra-Terminal (BET) Degraders Derived from Triazolodiazepine (JQ1) and Tetrahydroquinoline (I-BET726) BET Inhibitor Scaffolds

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Authors: Kwok-Ho Chan, Michael Zengerle, Andrea Testa, Alessio Ciulli

Journal title: Journal of Medicinal Chemistry

Journal publisher: American Chemical Society

Published year: 2017

DOI identifier: 10.1021/acs.jmedchem.6b01912

ISSN: 0022-2623