ERD

Epigenetic Drug Discovery

Project: EPITOOLS

Updated at: 27-04-2024

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Project acronym EPITOOLS

Highly selective inhibition of histone demethylases by de novo macrocyclic peptides

Project: EPITOOLS

Updated at: 27-04-2024

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Project acronym EPITOOLS

Structure-activity studies of a macrocyclic peptide inhibitor of histone lysine demethylase 4A

Project: EPITOOLS

Updated at: 27-04-2024

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Project acronym EPITOOLS

Investigating d -lysine stereochemistry for epigenetic methylation, demethylation and recognition

Project: EPITOOLS

Updated at: 27-04-2024

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Project acronym EPITOOLS

Investigations on small molecule inhibitors targeting the histone H3K4 tri-methyllysine binding PHD-finger of JmjC histo...

Project: EPITOOLS

Updated at: 27-04-2024

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Project acronym EPITOOLS

Non-competitive cyclic peptides for targeting enzyme–substrate complexes

Project: EPITOOLS

Updated at: 27-04-2024

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Project acronym EPITOOLS

Thioether Macrocyclic Peptides Selected against TET1 Compact Catalytic Domain Inhibit TET1 Catalytic Activity

Project: EPITOOLS

Updated at: 27-04-2024

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Project acronym EPITOOLS

Mechanistic and structural studies of KDM-catalysed demethylation of histone 1 isotype 4 at lysine 26

Project: EPITOOLS

Updated at: 27-04-2024

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Project acronym EPITOOLS

Use of cyclic peptides to induce crystallization: case study with prolyl hydroxylase domain 2

Project: EPITOOLS

Updated at: 27-04-2024

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Project acronym EPITOOLS

Periodic Reporting for period 4 - EPITOOLS (Chemical biology approaches to unraveling the histone code)

Project: EPITOOLS

Updated at: 27-04-2024

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Project acronym EPITOOLS

CHAPTER 5. Cyclic Peptides as Chemical Probes

Project: EPITOOLS

Updated at: 27-04-2024

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Project acronym EPITOOLS

Chemical Compounds Targeting DNA Methylation and Hydroxymethylation

Project: EPITOOLS

Updated at: 27-04-2024

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Project acronym EPITOOLS

Inhibitors of JmjC-Containing Histone Demethylases

Project: EPITOOLS

Updated at: 27-04-2024

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Project acronym EPITOOLS

Editorial overview: Epigenetics equals chemical biology

Project: EPITOOLS

Updated at: 27-04-2024

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Project acronym EPITOOLS

Structural diversity in de novo cyclic peptide ligands from genetically encoded library technologies

Project: EPITOOLS

Updated at: 27-04-2024

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Project acronym EPITOOLS

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Epigenetic Drug Discovery

Highly selective inhibition of histone demethylases by de novo macrocyclic peptides

Structure-activity studies of a macrocyclic peptide inhibitor of histone lysine demethylase 4A

Investigating d -lysine stereochemistry for epigenetic methylation, demethylation and recognition

Investigations on small molecule inhibitors targeting the histone H3K4 tri-methyllysine binding PHD-finger of JmjC histo...

Non-competitive cyclic peptides for targeting enzyme–substrate complexes

Thioether Macrocyclic Peptides Selected against TET1 Compact Catalytic Domain Inhibit TET1 Catalytic Activity

Mechanistic and structural studies of KDM-catalysed demethylation of histone 1 isotype 4 at lysine 26

Use of cyclic peptides to induce crystallization: case study with prolyl hydroxylase domain 2

Periodic Reporting for period 4 - EPITOOLS (Chemical biology approaches to unraveling the histone code)

CHAPTER 5. Cyclic Peptides as Chemical Probes

Chemical Compounds Targeting DNA Methylation and Hydroxymethylation

Inhibitors of JmjC-Containing Histone Demethylases

Editorial overview: Epigenetics equals chemical biology

Structural diversity in de novo cyclic peptide ligands from genetically encoded library technologies